NoteEnhanced solubility and antibacterial activity of lipophilic fluoro-substituted N-benzoyl-2-aminobenzothiazoles by complexation with β-cyclodextrins
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2019, Carbohydrate PolymersCitation Excerpt :Such literature suggestion is confirmed by our findings in the case of the S-unsubstituted benzothiazole compound 2 but not with 1. An important objective of this work was to gain information on the possible mechanism(s) of antibacterial activity enhancement after complexation with CDs and, in this regard, several proposals have been made (Athanassiou et al., 2003; Trapani et al., 2016) which essentially focus on two aspects. The first one is the improvement of dissolution properties arising from the complexation with CDs.
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