Abstract
A method for the preparation ofN-monoacyl imidazolidines and hexahydropyrimidines (as hydrochlorides) by interaction of monoacylated derivatives of ethylenediamine and trimethylenediamine with chloromethyl methyl ether was developed. Also a method for the preparation ofN,N′-diacylimidazolidines and hexahydropyrimidines either by acylation of their monoacyl derivatives or by reaction of the correspondingN,N′-diacyl alkylenediamine derivatives with dimethoxymethane, diacetoxymethane, 1,3,5-trioxane or chloromethyl methyl ether was designed.
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Translated fromIzvestiya Akademii Nauk. Seriya Khimicheskaya, No. 8, pp. 1452–1456, August, 1994.
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Luk'yanov, O.A., Pokhvisneva, G.V. & Ternikova, T.V. N,N′-Diacylated imidazolidines and hexahydropyrimidines. Russ Chem Bull 43, 1376–1380 (1994). https://doi.org/10.1007/BF00703698
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DOI: https://doi.org/10.1007/BF00703698